Some of the Peptides
How does Sermorelin work?
Sermorelin is a synthetic hormone peptide similar in structure to a growth hormone releasing hormone (GHRH). It’s commonly utilized to optimize growth hormone levels in adults, offering a variable IGF-1 increase.
Sermorelin works to burn fat, increase lean muscle, improve hormonal balance, enhance energy and boost the immune system.
How does Glycine work?
Glycine is an amino acid that can also act as a neurotransmitter. It has been used to help treat BPH, schizophrenia, and stroke. Research has shown that it can also help to stimulate the pituitary gland to secrete growth hormone without increasing prolactin levels. Glycine plays an important role in the control of the hypothalamic-pituitary function, specifically impacting growth hormone release. Glycine is an amino acid that acts as a stimulatory agent inducing the pituitary gland to secrete hGH.
Glycine goes far beyond encouraging weight loss and enhancing lean muscle mass. Enjoy a better night’s sleep, less mental daytime fatigue, enhance mental clarity/cognition, significantly improved skin elasticity, tone and texture, while receiving an enhanced synergistic boost to IGF-
Thymosin Alpha-1 is a major component of Thymosin Fraction 5 found in the thymus. The thymus is responsible for regulating the immune system. Thymosin Alpha-1 is prescribed to optimize the performance of your immune health and improve general wellness by preventing infections such as the common cold or the flu. It acts to augment T-cell function; T-cells are a part of the adaptive immune system which fights off infection. It is best prescribed to be taken once daily until vial is empty.
How does Thymosin Alpha-1 work?
T-cells come in two forms: killer and helper cells. Killer T-cells are responsible for hunting down and destroying our body’s own cells that are cancerous or infected with bacteria or viruses. TA-1 is thought to modulate the immune system by augmenting T-cell function. TA-1 may affect thymocytes by stimulating their differentiation or by converting them to active T-cells.
What forms of Thymosin Alpha-1 are available?
TA-1 is available reconstituted for subcutaneous injection.
What you need to know about Thymosin Alpha-1
Thymosin Alpha-1 appears to be well tolerated. No adverse drug interaction has been observed. No side effects, other than some irritation or burning sensation at the site of injection, have been reported.
Benefits of Thymosin Alpha-1
Thymosin Alpha-1 has been shown to exhibit antibacterial, antiviral, and antifungal properties, increase vaccine effectiveness, suppress tumor growth, enhance the function of certain immune cells, help eradicate unhealthy cells, stop infection or cancer growth, strengthen your immune system, and improve symptoms associated with chronic fatigue.
Thymosin Beta-4 has been found to play an important role in protection, regeneration, and remodeling on injured or damaged tissue. Thymosin is a hormone secreted from the thymus. The thymus is responsible for regulating the immune system and tissue repair. Thymosin Beta-4 is prescribed for acute injury, surgical repair, and patients that were once athletes and accumulated injuries over time. It acts as a major actin-sequestering molecule and can be taken after cardiac injury for better healing of the tissue in the heart. It is best prescribed to be taken once daily for 20 days.
How does Thymosin Beta-4 work?
Thymosin Beta-4 is typically found in both types of muscle in the human body – skeletal (the muscles that are required to move) and smooth (muscles such as those in the heart). When damage to the tissue occurs, Thymosin Beta-4 is upregulated. It is released in the body to help people heal from traumas. In the process of healing from injury, it also acts to reduce the amount of scar tissue and improve flexibility. It also has potent anti-inflammatory properties. Its primary function is to stimulate the production of T cells, which are an important part of the immune system. Thymosin also assists in the development of B cells to plasma cells to produce antibodies. Thymosin Beta-4 is a member of a highly conserved family of actin monomer-sequestering proteins. In addition to its role as a major actin-sequestering molecule, Thymosin Beta-4 has a role in tissue repair.
Benefits of Thymosin Beta-4
Thymosin Beta-4 has been shown to calm muscle spasms, improve muscle tone, increase exchange of substances between cells, encourage tissue repair, help maintain flexibility, reduce inflammation of tissue in joints, encourage the growth of new blood cells in tissue, increase endurance and strength, and prevent the formation of adhesions and fibrous bands in muscles, tendons, and ligaments.
Pentosan Polysulfate is a semi-synthetic polysulfated xylan used for the relief of Osteoarthritis. The mechanism of PPS action in osteoarthritis is multifactorial, with both stimulation of cartilage matrix synthesis and the prevention of cartilage breakdown. There are also systemic effects on blood lipid and fibrinolysis that may help clear the subchondral circulation. This is mainly used for osteoarthritis and inflammatory related skeletal conditions.
How does Pentosan Polysulfate work?
In one study, after a series of four to six intra-articular PPS injections into the knees of human volunteers, there was a significant increase in the size of the synovial fluid hyaluronan without causing any inflammation or bleeding into the joint cavity.
Benefits of Pentosan Polysulfate
Pentosan Polysulfate has been shown to reduce inflammation, optimize peptides, help with osteoarthritis, stimulate cartilage matrix synthesis and the prevention of cartilage, and it has anti-thrombotic properties. It has systemic effects on blood lipid and fibrinolysis that may help clear the subchondral circulation.
Bremelanotide PT-141 was developed from the peptide hormone Melanotan II for aphrodisiac effects. Bremelanotide PT-141 effects sexual function via interaction with the hypothalamus. Its usage has been found to increase erection in 80% of males who did not respond to Viagra or Cialis. Bremelanotide PT-141 has all shown an ability to increase the chances of women achieving at least one sexually gratifying experience by up to 50%.
How does Bremelanotide PT-141 work?
Unlike other sexual enhancement drugs, Bremelanotide PT-141 acts at the level of the brain, thus eliciting a rather natural sexual response. Melanotan II is a peptide hormone that acts to increase sexual arousal by interacting with the hypothalamus in the brain. As a derivative of MT-II, Bremelanotide PT-141 induces sexual arousal by binding to melanocortin receptors in the hypothalamus.
What you need to know about Bremelanotide PT-141:
Reported side effects of Bremelanotide PT-141 are flushing, nausea, and gastrointestinal upset. No contraindications have been reported.
Benefits of Bremelanotide PT-141
Bremelanotide PT-141 has been shown to produce rapid onset of sexual arousal, heightened libido, improve symptoms of female sexual dysfunction, induce erection in men suffering from ED, and improve sexual dysfunction on the level of the central nervous system. Bremelanotide PT-141 is available for subcutaneous injection.
BPC-157 is a partial sequence of body protection compound (BPC) found in human gastric juice. It can be used to accelerate healing of a variety of wounds including tendon-to-bone healing and the healing of damaged ligaments. It acts systematically in the digestive tract to combat leaky gut, IBS, gastrointestinal cramps and Crohn’s disease. BPC-157 protects and prevents gastric ulcers. It can be used to protect the liver from toxic damage (alcohol, antibiotics, etc.). Lastly, it promotes healing of traumatic brain injury (TBI).
How does BPC-157 work?
In response to tendon and ligament injury, BPC-157 accelerates healing by increasing type 1 collagen in these tissues. BPC-157 is cytoprotective and thus helps maintain the mucosal lining of the GI tract. As an anti-inflammatory, it aids in the protection and healing of inflamed intestinal issues. Additionally, BPC-157 acts as a neuroprotective by modulating serotonin and dopamine production in the brain.
What you need to know about BPC-157:
BPC-157 is a stable gastric peptide and has been found as a safe treatment for inflammatory bowel disease, ligament wounds and tendon-to-bone wounds. It is a stable human gastric juice and has no reported toxicity.
What forms of BPC-157 are available?
BPC-157 is available as a subcutaneous injection and as an oral capsule.
Benefits of BPC-157
BPC-157 has shown improved healing of many types of wounds, protect intestinal organs and prevent leaky stomach ulcers, combat leaky gut, IBS, gastrointestinal cramps and Crohn’s disease, accelerate healing of skin burns, anti-inflammatory, maintain an integrity of mucosal lining in GI tract, repair tissues of GIT, tendons, ligaments, brain, bone, etc., improve digestive function, and protect and promote healing of liver due to toxic stress.
Melanotan I and Melanotan II are both analogs of the peptide hormone alpha-melanocyte- stimulating hormone (a-MSH) that induces skin tanning. Like its predecessor, Melanotan I, MT-II plays a role in stimulating melanogenesis and thus provides a protective mechanism against UV rays, since under its actions, melanocytes are able to increase production and secretion of the hormone melanin. Scientists have also noticed that MT 2 had a positive effect on libido due to its aphrodisiac properties. Additionally, MT 2 exhibits a mild positive fat-mobilizing effects. Melanotan I is an FDA approved drug under the brand name Scenesse. Scenesse is most used to treat patients that have an intolerance to light.
A pilot phase I study was conducted with a cyclic heptapeptide analog of alpha-melanocyte stimulating hormone (alpha MSH). The lactam-bridged molecule, called Melanotan II (MT-II), has the structure of AC-Nle4-Asp5-His6-DPhe7-Arg8-Trp9-Lys10 alpha-MSH4-10-NH2 (MT-II) and has super potent melanotropic activity in vitro. A single-blind, alternating day (saline or MT-II), placebo-controlled trial was conducted in 3 normal male volunteers starting at the dose of 0.01 mg/kg of MT-II. Subcutaneous injections of MT-II or saline were given daily (Monday-Friday) for 2 consecutive weeks. Two subjects were escalated by 0.005 mg/kg increments to 0.03 mg/kg and one to 0.025 mg/kg. The 0.03 mg/kg dose produced Grade II somnolence and fatigue in one of two subjects (WHO standards). Mild nausea, not requiring antiemetic treatment, was reported at more MT-II dose levels. A stretching and yawning complex appeared to correlate with the onset of spontaneous, Penile erections which were intermittently experienced for 1-5 hours after MT-II dosing, depending on the MT-II dose. Two subjects had increased pigmentation in the fact, upper body, and buttock, as measured by quantitative reflectance and by visual perception 1 week after MT-II dosing ended. These results demonstrate that MT-II has tanning activity in humans given only 5 low dose every other day by subcutaneous injection. The recommended single MT-II dose for future Phase I studies is 0.025 mg/kg / day.
Melanotan I FAQs
· What is Melanotan I?
Melanotan I and Melanotan II are both analogs of the peptide hormone alpha-melanocyte-stimulating hormone (a-MSH) that induces skin tanning. Like its predecessor, Melanotan I, MT-II plays a role in stimulating melanogenesis. Thus, it provides a protective mechanism against UV rays since, under its actions, melanocytes are able to increase production and secretion of the hormone melanin. Scientists also noticed that MT-II had a positive effect on libido due to its aphrodisiac properties. Additionally, MT-II exhibits a mild fat-mobilizing effect. Melanotan I is an FDA approved drug under the brand name Scenesse, which is most commonly used to treat patients that have an intolerance to light.
· What can Melanotan I help with?
Melanotan I plays a prominent role in the production of pigment in the skin that allows for self-tanning with lower UV exposure. This means that the body will grow tanned all over, even in places that aren’t exposed to sunlight. However, UV exposure will accelerate the tanning process in exposed areas. It also helps reduce sun damage and increases sexual arousal, sexual desire, and appetite.
· What is the recommended dosing schedule?
Inject 0.15 mL once daily for 1-2 weeks then 0.25 mL twice weekly after that for maintenance.
· Are there any side effects?
Melanotan I is generally considered to be milder than Melanotan II. Studies have shown that Melanotan I can take much longer to develop than Melanotan II. Other side effects of this formula include facial flushing, nausea, and new or darkened freckles.
· Can this product be taken by a pregnant women or women who are nursing?
It is not recommended that this product be taken by those who are pregnant or nursing without consulting a medical professional first.
· Can men and women take this product?
Melanotan I can be consumed by men and women.
· Where is this product made/manufactured?
All medications are compounded in house at Tailor Made Compounding in the United States. Tailor Made Compounding 503A compounding pharmacy outfitted with two USP 795 Non-Sterile compounding facilities, three USP 797 Sterile compounding facilities, and one USP 800 Hazardous Sterile compounding facility.